Asset profile

Budesonide (targeted-release) · TARPEYO / Nefecon

Small molecule

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Approvedregulatory verdict

Evidence outlook

Approved: Chronic Kidney Disease, Primary IgA Nephropathy

Regulatory approval supersedes design-level evidence grading; the trials behind approval are preserved below as the drug's evidence history.

track record: Reliable signal

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Competitive landscape

80 competitors in this universe: 1 direct rival (same mechanism and indication), 19 same-class, 60 same-indication.

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DrugStageModalityMechanismEvidence signalReported efficacygraded featured trials
Budesonide (targeted-Release) (TARPEYO / Nefecon): this drugApprovedSmall moleculeGlucocorticoid receptor
Relacorilant (Lifyorli)ApprovedSmall moleculeGlucocorticoid receptor
Albuterol / Budesonide (Airsupra)ApprovedCombinationBeta-2 adrenergic receptor, Glucocorticoid receptor, Glucocorticoid receptor / Beta-2 adrenergic receptor
Beclomethasone (QVAR)ApprovedSmall moleculeGlucocorticoid receptor
Budesonide (Entocort EC)Approved—Glucocorticoid receptor
Budesonide (Ortikos)Approved—Glucocorticoid receptor
Budesonide (Uceris Rectal Foam)Approved—Glucocorticoid receptor
Budesonide MMX (Uceris)Approved—Glucocorticoid receptor
Ciclesonide (Alvesco)ApprovedSmall moleculeGlucocorticoid receptor
Fluticasone FuroateApprovedSmall moleculeGlucocorticoid receptor
Fluticasone Furoate / Umeclidinium / Vilanterol (Trelegy Ellipta)ApprovedSmall moleculeMuscarinic acetylcholine receptor (M3), Beta-2 adrenergic receptor, Glucocorticoid receptor, Glucocorticoid receptor / Beta-2 adrenergic receptor / Muscarinic M3 receptor (ICS/LABA/LAMA triple combination)
Fluticasone Furoate / VilanterolApprovedSmall moleculeBeta-2 adrenergic receptor, Glucocorticoid receptor, Glucocorticoid receptor / Beta-2 adrenergic receptor
Fluticasone PropionateApprovedSmall moleculeGlucocorticoid receptor
Fluticasone Propionate / Salmeterol (Advair HFA)ApprovedCombinationGlucocorticoid receptor, Beta-2 adrenergic receptor, Glucocorticoid receptor / Beta-2 adrenergic receptor
Halobetasol Propionate Foam (Lexette)ApprovedSmall moleculeGlucocorticoid receptor
Halobetasol Propionate Lotion (Bryhali)ApprovedSmall moleculeGlucocorticoid receptor

…and 65 more. Research shows the complete landscape.

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Research adds each competitor's evidence grade and sourced trial results, aligned per race, so you can see who actually has the data.

Upcoming events

(4 total)

Estimated primary-completion dates from ClinicalTrials.gov. These are registry estimates, never confirmed readout dates; they can move as trials progress.

2026 (2)
December 2026 (2)
Phase 4Glomerulonephritis, IGA, Probiotics, BudesonideNot yet recruiting
Est. primary completion 2026-12-31 · NCT06528015 · CT.gov ↗
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Phase 4Chronic Kidney DiseaseRecruiting
Est. primary completion 2026-12-31 · NCT07030894 · CT.gov ↗
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2027 (1)
March 2027 (1)
Phase 4Chronic Kidney DiseaseActive not recruiting
Est. primary completion 2027-03 · NCT06712407 · CT.gov ↗
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2029 (1)
August 2029 (1)
Phase 4Chronic Kidney DiseaseRecruiting
Est. primary completion 2029-08 · NCT06676384 · CT.gov ↗
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See the full readout calendar ↗

All registered studies

Every ClinicalTrials.gov study of this drug's own program, grouped by indication and phase. Research unlocks the studies themselves: titles, statuses, dates and featured-trial cross-links.

Phase 3 (3)
Phase 1 (1)
Phase 4 (4)