Mechanism

JAK1 / JAK3 (with lesser JAK2 activity); metformin arm targets AMPK/hepatic gluconeogenesis

Assets acting on this target.

Class
Combination regimen: JAK inhibitor (tofacitinib/CP-690,550) plus metformin (biguanide, not itself an RA drug)
Pathway
Tofacitinib blocks JAK-STAT cytokine signaling; metformin studied as an adjunct via AMPK activation
Research

Explore this mechanism at different depths

Research adds deeper and simplified explanation variants while preserving the same scientific register and source caveats.

Company

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